"Keillor TG2 Inhibitors" (acrylamide compounds)

Keillor inhibitor AA9

Quantity Unit Price Status
10 mg 400 € Available
Documents
Art. No.
Z015
Synonym
CAS 2134114-20-6
Molecular Formula
C32H36N4O5
Molecular Weight
556.65
Purity by HPLC
>95 % (214 nm)
Appearance
White solid
Solubility
500 μM in 5% (v/v) DMSO / aqueous buffers.
DMSO stock solutions can be stored at -20°C for at least 6 months. To avoid too many freeze-thaw cycles, we strongly recommend storage of aliquots.
Application
Site specific inhibitor of tissue transglutaminase
KI = 9 μM; kinact/KI = 0.10 μM-1min-1 [1]
Storage
Store at -20°C, desiccate, keep away from light.
Reference(s)
[1] A. Akbar et al. J. Med. Chem. 2017, 60 (18), 7910–7927.
Note
INTENDED FOR RESEARCH USE ONLY, NOT FOR USE IN HUMAN, THERAPEUTIC OR DIAGNOSTIC APPLICATIONS.

News

Blog

Events