"Keillor TG2 Inhibitors" (acrylamide compounds)

Keillor inhibitor NC9

Quantity Unit Price Status
10 mg 400 € Available
Documents
Art. No.
Z016
Synonym
CAS 1352090-52-8
Molecular Formula
C35H47N5O8S
Molecular Weight
697.84
Purity by HPLC
>95 % (214 nm)
Appearance
Yellow, fluorescent solid
Solubility
100 μM in 5% (v/v) DMSO / aqueous buffers.
DMSO stock solutions can be stored at -20°C for at least 6 months. To avoid too many freeze-thaw cycles, we strongly recommend storage of aliquots.
Application
Site specific inhibitor of tissue transglutaminase
KI = 34 μM; kinact/KI = 0.08 μM-1min-1 [1]
Storage
Store at -20°C, desiccate, keep away from light.
Reference(s)
[1] A. Akbar et al. J. Med. Chem. 2017, 60 (18), 7910–7927.
Note
INTENDED FOR RESEARCH USE ONLY, NOT FOR USE IN HUMAN, THERAPEUTIC OR DIAGNOSTIC APPLICATIONS.

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