"Keillor TG2 Inhibitors" (acrylamide compounds)

Keillor inhibitor VA4

Quantity Unit Price Status
10 mg 400 € Available
Documents
Art. No.
Z017
Synonym
CAS 2088001-23-2
Molecular Formula
C33H41N5O6S
Molecular Weight
635.77
Purity by HPLC
>95 % (214 nm)
Appearance
Yellow, fluorescent solid
Solubility
100 μM in 20% (v/v) DMSO / aqueous buffers.
DMSO stock solutions can be stored at -20°C for at least 6 months. To avoid too many freeze-thaw cycles, we strongly recommend storage of aliquots.
Application
Site specific inhibitor of tissue transglutaminase
KI = 13 μM; kinact/KI = 0.11 μM-1min-1 [1]
Storage
Store at -20°C, desiccate, keep away from light.
Reference(s)
[1] A. Akbar et al. J. Med. Chem. 2017, 60 (18), 7910–7927.
Note
INTENDED FOR RESEARCH USE ONLY, NOT FOR USE IN HUMAN, THERAPEUTIC OR DIAGNOSTIC APPLICATIONS.

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