"Keillor TG2 Inhibitors" (acrylamide compounds)

Keillor inhibitor AA9



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10 mg 385 € available


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Art. No. Z015
Synonym CAS 2134114-20-6
Molecular Formula C32H36N4O5
Molecular Weight 556.65
Purity by HPLC >95 % (214 nm)
Appearance White solid
Solubility 500 μM in 5% (v/v) DMSO / aqueous buffers.
DMSO stock solutions can be stored at -20°C for at least 6 months. To avoid too many freeze-thaw cycles, we strongly recommend storage of aliquots.
Application Site specific inhibitor of tissue transglutaminase
KI = 9 μM; kinact/KI = 0.10 μM-1min-1 [1]
Storage Store at -20°C, desiccate, keep away from light.
Reference(s) [1] A. Akbar et al. J. Med. Chem. 2017, 60 (18), 7910–7927.
Note INTENDED FOR RESEARCH USE ONLY, NOT FOR USE IN HUMAN, THERAPEUTIC OR DIAGNOSTIC APPLICATIONS.

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